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期刊论文

Comparison of bronchodilating and anti-inflammatory activities of oral formoterol and its (R,R)-enantiomersl

陈季强XIE Qiang-Min CHEN Ji-Qiang SHEN Wen-Hui YANG Qiu-Huo BIAN Ru-Lian

Xie QM et a l/Acta Pharmacol Sin 2003 Mar; 24 (3): 277-282,-0001,():

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摘要/描述

To compare the bronchodilating and antiinflammatory effects of oral racemic formoterol (rac-FMT) and (R,R)-formoterol (R,R-FMT). METHODS: The changes of lung resistance (RL), dynamic lung compliance (Cdyn), and the accumulation of inflammatory cells in bronchoalveolar lavage fluids (BALF) induced by ovalbumin aerosol in sensitized guinea pigs and mice were investigated in vivo. RESULTS: Mean value increase of RL and mean value reduction of Cdyn from 1 to 30 min after antigen challenge were up to 101%

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